O. E. Jensen, S. O. Lawesson, R. Bardi, A. M. Piazzesi, and C. Toniolo, Studies on amino acids and peptides VIII, Tetrahedron, vol.41, issue.23, p.5595, 1985.
DOI : 10.1016/S0040-4020(01)91361-4

C. Mannich and W. Krosche, Ueber ein Kondensationsprodukt aus Formaldehyd, Ammoniak und Antipyrin, Archiv der Pharmazie, vol.15, issue.1, p.647, 1912.
DOI : 10.1002/ardp.19122500151

I. Ugi and R. Meyr, Neue Darstellungsmethode f??r Isonitrile, Angewandte Chemie, vol.63, issue.22-23, p.702, 1958.
DOI : 10.1002/ange.19580702213

W. P. Weber, G. W. Gokel, and I. Ugi, Phasen??bergangs-Katalyse bei der Hofmannschen Carbylamin-Reaktion, Angewandte Chemie, vol.4, issue.12, p.587, 1972.
DOI : 10.1002/ange.19720841211

P. Hoffmann, G. Gokel, D. Marquading, and I. , Ugi in Isonitrile Chemistry Academic press, c) I.A. O'Neil in Comprehensive Organic Functional Group Transformations, pp.1315-963, 1971.

Y. Kobayashi and T. Fukuyama, Development of a novel indole synthesis and its application to natural products synthesis, Journal of Heterocyclic Chemistry, vol.119, issue.5, p.1043, 1998.
DOI : 10.1002/jhet.5570350504

I. I. Hoffmann, S. Ugi, and R. Lohberger, Karl in Comprehensive Organic Synthesis, Pergamon : Oxford, 1991, 2, 1083. c) A. Dömling, I. Ugi, Angew. Chem. Int. Ed. Engl. Acc. Chem. Res, vol.133, issue.39, pp.3169-3198, 1971.

. Chem, C. Int, V. Hulme, and . Gore, 21, 810. g) I. Ugi, A. Dömling in Combinatorial Chemistry-A Practical Approach, Eur. J. Org. Chem. Curr. Med. Chem, vol.287, issue.10, p.51, 1133.

. Opin, 306. k) I. Ugi, A. Dömling, Chem. Biol. Comb. Chem, vol.6, issue.287, 2000.

. Dömling, 1. p) The Passerini Reaction L, Chem. Rev. Banfi, R. Riva in Organic Reactions, vol.106, issue.65, 2005.

T. Carofiglio, C. Floriani, A. Chiesi-villa, and C. Guastini, Isocyanide complexes of titanium(IV) and vanadium(V): concerning the nonexistent insertion of isocyanides into a metal-chloride bond, Inorganic Chemistry, vol.28, issue.24, pp.4417-1659, 1989.
DOI : 10.1021/ic00323a026

P. G. Carofiglio, C. Cozzi, A. Floriani, C. Chiesi-villa, and . Rizzoli, Nonorganometallic pathway of the Passerini reaction assisted by titanium tetrachloride, Organometallics, vol.12, issue.7, p.2726, 1993.
DOI : 10.1021/om00031a047

W. Mcfarland, Reactions of Cyclohexylisonitrile and Isobutyraldehyde with Various Nucleophiles and Catalysts, The Journal of Organic Chemistry, vol.28, issue.9, p.2179, 1963.
DOI : 10.1021/jo01044a006

R. Neidlein, I. Ugi, and F. K. , 43. a), Chem. Ber. Chem. Ber, vol.94, issue.110, pp.2233-1603, 1159.

J. W. Mcfarland, Reactions of Cyclohexylisonitrile and Isobutyraldehyde with Various Nucleophiles and Catalysts, The Journal of Organic Chemistry, vol.28, issue.9, p.2179, 1963.
DOI : 10.1021/jo01044a006

I. Chem, F. Ugi, L. Bodesheim, G. Ann, and W. Zinner, 163. 50. a), Chem. Arch. Pharm. Arch. Pharm, vol.652, issue.306, pp.61-94, 1962.

P. Hoffmann, G. Gokel, D. Marquarding, and I. , Ugi in Isonitrile Chemistry, p.9, 1971.

I. Ugi, F. K. Rosendahl, F. Bodesheim, and L. Ann, Chem. 1963, 666, 54. 57. a) I. Ugi, F. Bodesheim, Liebigs Ann, Chem, vol.666, p.61, 1963.

S. B. Keum, D. H. Kang, H. Y. Lee, Y. Koh, and . Kim, An Efficient Synthesis of Morpholin-2-one Derivatives Using Glycolaldehyde Dimer by the Ugi Multicomponent Reaction, Organic Letters, vol.3, issue.26, p.4149, 2001.
DOI : 10.1021/ol016716w

A. Failli, H. Immer, and M. Götz, The synthesis of cyclic peptides by the four component condensation (4 CC), Canadian Journal of Chemistry, vol.57, issue.24, p.3257, 1979.
DOI : 10.1139/v79-533

D. Bonne, M. Dekhane, and J. Zhu, Modulating the Reactivity of ??-Isocyanoacetates: Multicomponent Synthesis of 5-Methoxyoxazoles and Furopyrrolones, Angewandte Chemie International Edition, vol.143, issue.14, p.2485, 2007.
DOI : 10.1002/anie.200605005
URL : https://hal.archives-ouvertes.fr/hal-00157605

K. Paulvannan and J. W. Jacobs, Preparation of tricyclic nitrogen heterocycles via intramolecular Diels-Alder reaction of furans, Tetrahedron, vol.55, issue.24, pp.7433-1851, 1999.
DOI : 10.1016/S0040-4020(99)00390-7

T. A. Keating and R. W. Armstrong, Postcondensation Modifications of Ugi Four-Component Condensation Products:?? 1-Isocyanocyclohexene as a Convertible Isocyanide. Mechanism of Conversion, Synthesis of Diverse Structures, and Demonstration of Resin Capture, Journal of the American Chemical Society, vol.118, issue.11, p.2574, 1996.
DOI : 10.1021/ja953868b

Z. Xiang, T. Luo, K. Lu, J. Cui, X. Shi et al., Concise Synthesis of Isoquinoline via the Ugi and Heck Reactions, Organic Letters, vol.6, issue.18, p.3155, 2004.
DOI : 10.1021/ol048791n

J. Cossy, C. Willis, V. Bellosta, L. M. Pourashraf, P. Delair et al., Saint-Jalmes, Synthesis, J. Org. Chem, pp.65-6966, 2000.

J. Gubin, J. Luccheti, J. Mahaux, D. Nisato, G. Rosseels et al., A novel class of calcium-entry blockers: the 1-[[4-(aminoalkoxy)phenyl]sulfonyl]indolizines, Journal of Medicinal Chemistry, vol.35, issue.6, p.981, 1992.
DOI : 10.1021/jm00084a002

S. Teklu, L. L. Gundersen, T. Larsen, K. E. Malterud, and F. Rise, Indolizine 1-sulfonates as potent inhibitors of 15-lipoxygenase from soybeans, Bioorganic & Medicinal Chemistry, vol.13, issue.9, p.3127, 2005.
DOI : 10.1016/j.bmc.2005.02.056

A. R. Katritzky, G. Qiu, B. Yang, and H. Y. He, ]isoquinolines via Benzotriazole Methodology, The Journal of Organic Chemistry, vol.64, issue.20, p.7618, 1999.
DOI : 10.1021/jo9906936

Y. Liu, Z. Song, and B. Yan, General and Direct Synthesis of 3-Aminoindolizines and Their Analogues via Pd/Cu-Catalyzed Sequential Cross-Coupling/Cycloisomerization Reactions, Organic Letters, vol.9, issue.3, p.409, 2007.
DOI : 10.1021/ol062766v

C. R. Smith, E. M. Bunelle, A. J. Rhodes, and R. Sarpong, Pt-Catalyzed Cyclization/1,2-Migration for the Synthesis of Indolizines, Pyrrolones, and Indolizinones, Organic Letters, vol.9, issue.6, p.1169, 2007.
DOI : 10.1021/ol0701971

H. Pauls and F. Kröhnke, Untersuchungen an 2-Chlorpyridinium-Salzen, III. Umsetzungen mit CH-aciden Verbindungen und ??bergang in Indolizine, Chemische Berichte, vol.43, issue.4, p.1294, 1977.
DOI : 10.1002/cber.19771100413

G. Seitz and R. Tegethoff, Synthese schwefelhaltiger, anellierter Indolizine durch intramolekulare [3+2]-Cycloaddition mit Pyridinium-methyliden, Archiv der Pharmazie, vol.124, issue.3, p.135, 1993.
DOI : 10.1002/ardp.19933260304

U. Bora, A. Saikia, and R. C. Boruah, A Novel Microwave-Mediated One-Pot Synthesis of Indolizines via a Three-Component Reaction, Organic Letters, vol.5, issue.4, p.435, 2003.
DOI : 10.1021/ol020238n

S. K. Heatcock, S. G. Davidson, M. A. Mills, and . Sanner, Daphniphyllum alkaloids. 10. Classical total synthesis of methyl homodaphniphyllate, The Journal of Organic Chemistry, vol.57, issue.9, p.2531, 1992.
DOI : 10.1021/jo00035a007

J. S. Magnus, A. Mendoza, M. Stamford, P. Ladlow, G. Willis et al., Nonoxidative coupling methodology for the synthesis of the antitumor bisindole alkaloid vinblastine and a lower-half analog: solvent effect on the stereochemistry of the crucial C-15/C-18' bond, Journal of the American Chemical Society, vol.114, issue.26, pp.10232-947, 1986.
DOI : 10.1021/ja00052a020

M. Ogata and H. Matsumoto, The Reaction of Amides with Diethylthiocarbamoyl Chloride: A New Procedure for the Preparation of Nitriles and Thioamides, HETEROCYCLES, vol.11, issue.1, p.139, 1978.
DOI : 10.3987/S(N)-1978-01-0139

J. J. Bodine and M. Kaloustian, An Efficient Conversion of N-Alkyllactams to N-Alkylthiolactams, Synthetic Communications, vol.7, issue.10, p.787, 1982.
DOI : 10.1080/00397918208061918

A. B. Charrette and M. Grenon, Mild Method for the Conversion of Amides to Thioamides, The Journal of Organic Chemistry, vol.68, issue.14, p.5792, 2003.
DOI : 10.1021/jo0344485

R. S. Varma and D. Kumar, Microwave-Accelerated Solvent-Free Synthesis of Thioketones, Thiolactones, Thioamides, Thionoesters, and Thioflavonoids, Organic Letters, vol.1, issue.5, p.697, 2000.
DOI : 10.1021/ol990629a

C. H. Wang, F. Y. Hwang, J. M. Horng, and C. T. Chen, A Novel Synthetic Scheme for 2-Ethylthioisonicotinamide, HETEROCYCLES, vol.12, issue.9, p.1191, 1979.
DOI : 10.3987/R-1979-09-1191

E. C. Taylor and J. A. Zoltewicz, A NEW SYNTHESIS OF ALIPHATIC AND AROMATIC THIOAMIDES FROM NITRILES, Journal of the American Chemical Society, vol.82, issue.10, p.2656, 1960.
DOI : 10.1021/ja01495a078

W. Walter, W. Rubach, and C. O. Meese, Alkylierungsreaktionen an Thioamiden, VI. Isolierung vonE- undZ-Thioimids??ureestern, Chemische Berichte, vol.7, issue.1, p.171, 1980.
DOI : 10.1002/cber.19801130118

:. W. Revue, J. Walter, and . Voss, The Chemistry of Amides, p.442, 1970.

H. Suter and H. Zutter, Studien ??ber Benzthiazole als eventuelle orale Antidiabetica, Helvetica Chimica Acta, vol.30, issue.7a, p.1084, 1967.
DOI : 10.1002/hlca.19670500415

C. J. Paget, K. Kisner, R. L. Stone, and D. C. Delong, Heterocyclic substituted ureas. II. Immunosuppressive and antiviral activity of benzothiazolyl- and benzoxazolylureas, Journal of Medicinal Chemistry, vol.12, issue.6, p.1016, 1969.
DOI : 10.1021/jm00306a011

S. Yoshida, S. Shiokawa, K. I. Kawano, T. Ito, H. Murakami et al., Receptor Partial Agonist for Treatment of Diarrhea-Predominant Irritable Bowel Syndrome, Journal of Medicinal Chemistry, vol.48, issue.22, pp.7075-65, 1993.
DOI : 10.1021/jm050209t