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1. , N. , 2. Cy, 3. Cy, . Cy et al., 08 (ddd, J = 14, 2.51 (s, 3H, H 4 ), 2.21 (ddd, J = 14.4, 11.1, 3.7 Hz, 1H, pp.296-299, 1994.

1. Hz, J. =. 3h, and H. Cy, 1H, H 8 ), 3.84-3.72 (m, 1H, H 12 ), 2.78 (dd, J = 15, pp.32714879-32714880, 2005.

5. and H. Ar, CDCl 3 ; 400 MHz) ? 10.90 (br s, 1H, NMR, vol.7, issue.8, pp.43-50

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J. Cy, 2. Cy, 1. Cy, 4. Cym, and 1. Cy, The mixture was stirred overnight at 80°C. The Ugi-Smiles product was obtained after in vacuo evaporation of the solvent and flash column chromatography Yellow oil Yield 37.5 % (510 mg) over three steps 1 H NMR (CDCl 3, After 10 min, 1 equiv. of triisopropyl phosphite was added. After 10 min, 2 mL of acetonitrile, 1 equiv MHz) ? 7.47 (d, J = 8.0 Hz, 1H, H 4 ), 7.39 (d, J = 1.5 Hz, 1H, H 1 ), 7.32 (dd, J = 8.0, 1.5 Hz, 1H 6.3 Hz, 2H, CH-Me 2 ), 4.31 (d, J = 6.1 Hz, 2H, H 6 ), 4.19 (q, pp.58-59, 2007.